Phase I trial of ftorafur combined with mitomycin C or methyl-CCNU in gastrointestinal cancers

Cancer Treat Rep. 1977 May-Jun;61(3):463-7.

Abstract

Twenty-five patients with disseminated gastrointestinal malignancies were treated in a phase I study with a combination of ftorafur and mitomycin C or florafur and methyl-CCNU. Most patients had been heavily treated previously. Gastrointestinal, central nervous system, and marrow toxicity were manageable. Tumor regression was noted in five of 25 patients. A large-scale phase II study in untreated patients with gastrointestinal malignancies appears indicated with a combination of these agents.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenocarcinoma / drug therapy*
  • Bone Marrow / drug effects
  • Drug Evaluation
  • Drug Therapy, Combination
  • Fluorouracil / analogs & derivatives*
  • Gastrointestinal Neoplasms / drug therapy*
  • Humans
  • Hypotension, Orthostatic / chemically induced
  • Mitomycins / adverse effects
  • Mitomycins / therapeutic use*
  • Nitrosourea Compounds / therapeutic use*
  • Remission, Spontaneous
  • Semustine / adverse effects
  • Semustine / therapeutic use*
  • Tegafur / adverse effects
  • Tegafur / therapeutic use*

Substances

  • Mitomycins
  • Nitrosourea Compounds
  • Semustine
  • Tegafur
  • Fluorouracil