Water-Gated Proton Transfer Dynamics in Respiratory Complex I

J Am Chem Soc. 2020 Aug 12;142(32):13718-13728. doi: 10.1021/jacs.0c02789. Epub 2020 Jul 30.

Abstract

The respiratory complex I transduces redox energy into an electrochemical proton gradient in aerobic respiratory chains, powering energy-requiring processes in the cell. However, despite recently resolved molecular structures, the mechanism of this gigantic enzyme remains poorly understood. By combining large-scale quantum and classical simulations with site-directed mutagenesis and biophysical experiments, we show here how the conformational state of buried ion-pairs and water molecules control the protonation dynamics in the membrane domain of complex I and establish evolutionary conserved long-range coupling elements. We suggest that an electrostatic wave propagates in forward and reverse directions across the 200 Å long membrane domain during enzyme turnover, without significant dissipation of energy. Our findings demonstrate molecular principles that enable efficient long-range proton-electron coupling (PCET) and how perturbation of this PCET machinery may lead to development of mitochondrial disease.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Density Functional Theory
  • Electron Transport Complex I / chemistry
  • Electron Transport Complex I / metabolism*
  • Molecular Dynamics Simulation*
  • Oxidation-Reduction
  • Protons*
  • Water / chemistry
  • Water / metabolism*

Substances

  • Protons
  • Water
  • Electron Transport Complex I