Peptide-Functionalized Hydrogels Modulate Integrin Expression and Stemness in Adult Human Epidermal Keratinocytes

Adv Biosyst. 2019 Oct;3(10):e1900022. doi: 10.1002/adbi.201900022. Epub 2019 Aug 23.

Abstract

The extracellular matrix (ECM) controls keratinocyte proliferation, migration, and differentiation through β-integrin signaling. Wound-healing research requires expanding cells in vitro while maintaining replicative capacity; however, early terminal differentiation under traditional culture conditions limits expansion. Here, a design of experiments approach identifies poly(ethylene glycol)-based hydrogel formulations with mechanical properties (elastic modulus, E = 20.9 ± 0.56 kPa) and bioactive peptide sequences that mimic the epidermal ECM. These hydrogels enable systematic investigation of the influence of cell-binding domains from fibronectin (RGDS), laminin (YIGSR), and collagen IV (HepIII) on keratinocyte stemness and β1 integrin expression. Quantification of 14-day keratin protein expression shows four hydrogels improve stemness compared to standard techniques. Three hydrogels increase β1 integrin expression, demonstrating a positive linear relationship between stemness and β1 integrin expression. Multifactorial statistical analysis predicts an optimal peptide combination ([RGDS] = 0.67 mm, [YIGSR] = 0.13 mm, and [HepIII] = 0.02 mm) for maintaining stemness in vitro. Best-performing hydrogels exhibit no decrease in Ki-67-positive cells compared to standards (15% decrease, day 7 to 14; p < 0.05, Tukey Test). These data demonstrate that precisely designed hydrogel biomaterials direct integrin expression and promote proliferation, improving the regenerative capability of cultured keratinocytes for basic science and translational work.

Keywords: extracellular matrix; hydrogels; keratinocytes; peptides; poly(ethylene glycol).

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adult
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Extracellular Matrix Proteins / chemistry
  • Extracellular Matrix Proteins / metabolism
  • Gene Expression / drug effects*
  • Humans
  • Hydrogels* / chemistry
  • Hydrogels* / pharmacology
  • Integrins* / analysis
  • Integrins* / genetics
  • Integrins* / metabolism
  • Keratinocytes* / cytology
  • Keratinocytes* / drug effects
  • Microscopy, Fluorescence
  • Peptides / chemistry
  • Peptides / pharmacology
  • Polyethylene Glycols / chemistry
  • Polyethylene Glycols / pharmacology
  • Stem Cells / cytology
  • Stem Cells / drug effects

Substances

  • Extracellular Matrix Proteins
  • Hydrogels
  • Integrins
  • Peptides
  • Polyethylene Glycols