Near-Infrared Light-Triggered Chlorine Radical (. Cl) Stress for Cancer Therapy

Angew Chem Int Ed Engl. 2020 Nov 16;59(47):21032-21040. doi: 10.1002/anie.202007434. Epub 2020 Sep 7.

Abstract

Free radicals with reactive chemical properties can fight tumors without causing drug resistance. Reactive oxygen species (ROS) has been widely used for cancer treatment, but regrettably, the common O2 and H2 O2 deficiency in tumors sets a severe barrier for sufficient ROS production, leading to unsatisfactory anticancer outcomes. Here, we construct a chlorine radical (. Cl) nano-generator with SiO2 -coated upconversion nanoparticles (UCNPs) on the inside and Ag0 /AgCl hetero-dots on the outside. Upon near-infrared (NIR) light irradiation, the short-wavelength emission UCNP catalyzes . Cl generation from Ag0 /AgCl with no dependence on O2 /H2 O2 . . Cl with strong oxidizing capacity and nucleophilicity can attack biomolecules in cancer cells more effectively than ROS. This . Cl stress treatment will no doubt broaden the family of oxidative stress-induced antitumor strategies by using non-oxygen free radicals, which is significant in the development of new anticancer agents.

Keywords: Ag0/AgCl hetero-dots; chlorine radicals; hypoxia; oxidative stress; upconversion nanoparticles.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / pharmacology*
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cell Survival / drug effects
  • Chlorine / chemistry
  • Chlorine / pharmacology*
  • Drug Screening Assays, Antitumor
  • Female
  • Free Radicals / chemistry
  • Free Radicals / pharmacology*
  • Infrared Rays
  • Mammary Neoplasms, Experimental / drug therapy
  • Mammary Neoplasms, Experimental / metabolism
  • Mammary Neoplasms, Experimental / pathology
  • Mice
  • Nanoparticles / chemistry
  • Oxidative Stress / drug effects
  • Particle Size
  • Photosensitizing Agents / chemistry
  • Photosensitizing Agents / pharmacology*
  • Silicon Dioxide / chemistry
  • Silicon Dioxide / pharmacology
  • Silver / chemistry
  • Silver / pharmacology
  • Surface Properties

Substances

  • Antineoplastic Agents
  • Free Radicals
  • Photosensitizing Agents
  • Silver
  • Chlorine
  • Silicon Dioxide