Transient receptor potential melastatin 2 contributes to neuroinflammation and negatively regulates cognitive outcomes in a pilocarpine-induced mouse model of epilepsy

Int Immunopharmacol. 2020 Oct:87:106824. doi: 10.1016/j.intimp.2020.106824. Epub 2020 Jul 27.

Abstract

Neuroinflammation contributes to the generation of epileptic seizures and is associate with neuropathology and comorbidities. Transient receptor potential melastatin 2 (TRPM2) expresses in various cell types in the brain. It plays a pathological role in a wide range of neuroinflammatory diseases, but has yet been studied in epilepsy. Here, a temporal lobe epilepsy model was generated by pilocarpine administration in mice. At 24 h, knockout (KO) TRPM2 alleviated the level of neuroinflammation, showing a reduction of IL-1β, TNF-α, CXCL2 and IL-6 mRNA production, NLRP3, ASC, and Caspase-1 protein expression and glial activation. Moreover, KO TRPM2 alleviated neurodegeneration, concurrent with reduced Beclin-1 and ATG5 protein expression. Later, KO TRPM2 ameliorated the epilepsy-induced psychological disorders, with improved performance in the open-field, Y maze and novel object recognition test. Together, these results suggest that TRPM2 facilitates epilepsy-related brain injury and may shed light on its potential as a therapeutic target for epilepsy-associated neuropathology and comorbidities.

Keywords: Autophagy; Cognitive impairment; Epilepsy; Neuroinflammation; Neuronal degeneration; TRPM2 ion channel.

MeSH terms

  • Animals
  • Behavior, Animal
  • Cognition*
  • Cytokines / genetics
  • Disease Models, Animal
  • Epilepsy* / chemically induced
  • Epilepsy* / genetics
  • Epilepsy* / metabolism
  • Epilepsy* / pathology
  • Hippocampus / metabolism
  • Hippocampus / pathology
  • Inflammation / genetics
  • Inflammation / metabolism
  • Inflammation / pathology
  • Male
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Neurons / pathology
  • Pilocarpine
  • TRPM Cation Channels* / genetics
  • TRPM Cation Channels* / metabolism

Substances

  • Cytokines
  • TRPM Cation Channels
  • TRPM2 protein, mouse
  • Pilocarpine