Parkinson's disease-related phosphorylation at Tyr39 rearranges α-synuclein amyloid fibril structure revealed by cryo-EM

Proc Natl Acad Sci U S A. 2020 Aug 18;117(33):20305-20315. doi: 10.1073/pnas.1922741117. Epub 2020 Jul 31.

Abstract

Posttranslational modifications (PTMs) of α-synuclein (α-syn), e.g., phosphorylation, play an important role in modulating α-syn pathology in Parkinson's disease (PD) and α-synucleinopathies. Accumulation of phosphorylated α-syn fibrils in Lewy bodies and Lewy neurites is the histological hallmark of these diseases. However, it is unclear how phosphorylation relates to α-syn pathology. Here, by combining chemical synthesis and bacterial expression, we obtained homogeneous α-syn fibrils with site-specific phosphorylation at Y39, which exhibits enhanced neuronal pathology in rat primary cortical neurons. We determined the cryo-electron microscopy (cryo-EM) structure of the pY39 α-syn fibril, which reveals a fold of α-syn with pY39 in the center of the fibril core forming an electrostatic interaction network with eight charged residues in the N-terminal region of α-syn. This structure composed of residues 1 to 100 represents the largest α-syn fibril core determined so far. This work provides structural understanding on the pathology of the pY39 α-syn fibril and highlights the importance of PTMs in defining the polymorphism and pathology of amyloid fibrils in neurodegenerative diseases.

Keywords: amyloid fibril structure; posttranslational modifications; α-synuclein.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amyloid / chemistry
  • Amyloid / metabolism
  • Animals
  • Cells, Cultured
  • Cryoelectron Microscopy
  • Gene Expression Regulation / drug effects
  • Humans
  • Models, Molecular
  • Neurons / drug effects
  • Neurons / metabolism
  • Parkinson Disease*
  • Phosphorylation
  • Protein Conformation
  • Rats
  • Rats, Sprague-Dawley
  • alpha-Synuclein / chemical synthesis
  • alpha-Synuclein / chemistry*
  • alpha-Synuclein / metabolism

Substances

  • Amyloid
  • alpha-Synuclein