Investigation on the Antibacterial Activity of Electronic Cigarette Liquids (ECLs): A Proof of Concept Study

Curr Pharm Biotechnol. 2021;22(7):983-994. doi: 10.2174/1389201021666200903121624.

Abstract

Background: The key ingredients of e-cigarettes liquid are commonly propane-1,2-diol (also called propylene glycol) and propane-1,2,3-triol (vegetal glycerol) and their antimicrobial effects are already established. The nicotine and flavors which are often present in e-liquids can interfere with the growth of some microorganisms.

Objective: The effect of combining these elements in e-liquids is unknown. The aim of the study was to investigate the possible effects of these liquids on bacterial growth in the presence or absence of nicotine and flavors.

Methods: Susceptibilities of pathogenic strains (Klebsiella pneumoniae, Staphylococcus aureus, Pseudomonas aeruginosa, Acinetobacter baumannii, Escherichia coli, Enterococcus faecalis and Sarcina lutea) were studied by means of a multidisciplinary approach. Cell viability and antioxidant assays were also evaluated.

Results: All e-liquids investigated showed antibacterial activity against at least one pathogenic strain. Higher activity was correlated to the presence of flavors and nicotine.

Discussion: In most cases, the value of minimal bactericidal concentration is equal to the value of minimal inhibitory concentration showing that these substances have a bactericidal effect. This effect was observed in concentrations up to 6.25% v/v. Antioxidant activity was also correlated to the presence of flavors. Over time, the viability assay in human epithelial lung A549 cells showed a dose-dependent inhibition of cell growth.

Conclusion: Our results have shown that flavors considerably enhance the antibacterial activity of propane-1,2-diol and propane-1,2,3-triol. This study provides important evidence that should be taken into consideration in further investigative approaches, to clarify the different sensitivity of the various bacterial species to e-liquids, including the respiratory microbiota, to highlight the possible role of flavors and nicotine.

Keywords: 2; 2-diol; 3-triol; Electronic cigarettes; antibacterial activity; e-liquids; flavors; nicotine; propane-1.

MeSH terms

  • A549 Cells
  • Anti-Bacterial Agents / pharmacology*
  • Cell Survival / drug effects
  • Cell Survival / physiology
  • Electronic Nicotine Delivery Systems*
  • Escherichia coli / drug effects
  • Escherichia coli / physiology
  • Flavoring Agents / pharmacology*
  • Glycerol / pharmacology*
  • Humans
  • Klebsiella pneumoniae / drug effects
  • Klebsiella pneumoniae / physiology
  • Microbial Sensitivity Tests / methods
  • Nicotine / pharmacology
  • Proof of Concept Study*
  • Propylene Glycol / pharmacology*
  • Pseudomonas aeruginosa / drug effects
  • Pseudomonas aeruginosa / physiology
  • Staphylococcus aureus / drug effects
  • Staphylococcus aureus / physiology

Substances

  • Anti-Bacterial Agents
  • Flavoring Agents
  • Propylene Glycol
  • Nicotine
  • Glycerol