An optimized acetylcholine sensor for monitoring in vivo cholinergic activity

Nat Methods. 2020 Nov;17(11):1139-1146. doi: 10.1038/s41592-020-0953-2. Epub 2020 Sep 28.

Abstract

The ability to directly measure acetylcholine (ACh) release is an essential step toward understanding its physiological function. Here we optimized the GRABACh (GPCR-activation-based ACh) sensor to achieve substantially improved sensitivity in ACh detection, as well as reduced downstream coupling to intracellular pathways. The improved version of the ACh sensor retains the subsecond response kinetics, physiologically relevant affinity and precise molecular specificity for ACh of its predecessor. Using this sensor, we revealed compartmental ACh signals in the olfactory center of transgenic flies in response to external stimuli including odor and body shock. Using fiber photometry recording and two-photon imaging, our ACh sensor also enabled sensitive detection of single-trial ACh dynamics in multiple brain regions in mice performing a variety of behaviors.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholine / metabolism*
  • Animals
  • Animals, Genetically Modified
  • Behavior, Animal / physiology
  • Biosensing Techniques / methods*
  • Brain / metabolism*
  • Cholinergic Agents / pharmacology
  • Drosophila / genetics
  • Drosophila / metabolism
  • Green Fluorescent Proteins / genetics
  • Green Fluorescent Proteins / metabolism
  • HEK293 Cells
  • Humans
  • Mice
  • Mushroom Bodies / metabolism
  • Neurons / metabolism
  • Olfactory Cortex / metabolism
  • Receptor, Muscarinic M3 / genetics
  • Receptor, Muscarinic M3 / metabolism
  • Somatosensory Cortex / metabolism

Substances

  • Cholinergic Agents
  • Receptor, Muscarinic M3
  • Green Fluorescent Proteins
  • Acetylcholine