Caffeine, exercise physiology, and time-trial performance: no effect of ADORA2A or CYP1A2 genotypes

Appl Physiol Nutr Metab. 2021 Jun;46(6):541-551. doi: 10.1139/apnm-2020-0551. Epub 2020 Nov 10.

Abstract

The aim of this study was to investigate the influence of ADORA2A and CYP1A2 genotypes on the physiological and ergogenic effects of caffeine. Sixty-six male cyclists were screened for ADORA2A and CYP1A2 genotypes; with 40 taking part subsequently in a randomised, double-blind, placebo-controlled study. Trial 1 was used to establish the oxygen uptake-power output relationship and maximal oxygen uptake. In trials 2 and 3, participants ingested 5 mg·kg-1 of caffeine or placebo 1 h before completing a submaximal incremental cycling test, followed by a time-trial (∼30 min). Relative to placebo, caffeine led to a significant reduction in time to complete the time-trial (caffeine: 29.7 ± 1.8 min; placebo: 30.8 ± 2.3 min); but there was no effect of genotype. During submaximal exercise, caffeine reduced mean heart rate by 2.9 ± 3.7 beats·min-1, with effects dissipating as exercise intensity increased. Caffeine also significantly reduced perceived exertion by 0.5 ± 0.8, and increased blood lactate by 0.29 ± 0.42 mmol·L-1, respiratory exchange ratio by 0.013 ± 0.032, and minute ventilation by 3.1 ± 6.8 L·min-1. Nonetheless, there were no supplement × genotype interactions. In conclusion, caffeine influences physiological responses to submaximal exercise and improves time-trial performance irrespective of ADORA2A or CYP1A2 genotypes. Novelty: Caffeine affects physiological responses at rest and during submaximal exercise independent of ADORA2A or CYP1A2 genotypes. Variability in the effect of caffeine on time-trial performance is not explained by ADORA2A or CYP1A2 genotypes.

Keywords: café; cardiorespiratoire; cardiorespiratory; coffee; cycling; cyclisme; endurance exercise; ergogenic; ergogène; exercice d’endurance; genetics; génétique.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Biomarkers / blood
  • Caffeine / administration & dosage*
  • Cytochrome P-450 CYP1A2 / genetics*
  • Double-Blind Method
  • Exercise / physiology*
  • Exercise Test
  • Genotype
  • Heart Rate / physiology
  • Humans
  • Lactates / blood
  • Male
  • Oxygen Consumption / physiology
  • Performance-Enhancing Substances / administration & dosage*
  • Physical Exertion / physiology
  • Receptor, Adenosine A2A / genetics*
  • Respiratory Function Tests

Substances

  • ADORA2A protein, human
  • Biomarkers
  • Lactates
  • Performance-Enhancing Substances
  • Receptor, Adenosine A2A
  • Caffeine
  • CYP1A2 protein, human
  • Cytochrome P-450 CYP1A2