D-mannose suppresses macrophage IL-1β production

Nat Commun. 2020 Dec 11;11(1):6343. doi: 10.1038/s41467-020-20164-6.

Abstract

D-mannose is a monosaccharide approximately a hundred times less abundant than glucose in human blood. Previous studies demonstrated that supraphysiological levels of D-mannose inhibit tumour growth and stimulate regulatory T cell differentiation. It is not known whether D-mannose metabolism affects the function of non-proliferative cells, such as inflammatory macrophages. Here, we show that D-mannose suppresses LPS-induced macrophage activation by impairing IL-1β production. In vivo, mannose administration improves survival in a mouse model of LPS-induced endotoxemia as well as decreases progression in a mouse model of DSS-induced colitis. Phosphomannose isomerase controls response of LPS-activated macrophages to D-mannose, which impairs glucose metabolism by raising intracellular mannose-6-phosphate levels. Such alterations result in the suppression of succinate-mediated HIF-1α activation, imposing a consequent reduction of LPS-induced Il1b expression. Disclosing an unrecognized metabolic hijack of macrophage activation, our study points towards safe D-mannose utilization as an effective intervention against inflammatory conditions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Differentiation / drug effects
  • Cell Line
  • Colitis / metabolism
  • Colitis / pathology
  • Gene Expression Regulation
  • Humans
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Inflammation / metabolism
  • Interleukin-1beta / genetics
  • Interleukin-1beta / metabolism*
  • Lipopolysaccharides / adverse effects
  • Macrophage Activation / drug effects*
  • Macrophages / drug effects*
  • Macrophages / metabolism*
  • Mannose / metabolism*
  • Mannose / pharmacology*
  • Mannosephosphates / metabolism
  • Metabolic Networks and Pathways / drug effects
  • Metabolomics
  • Monocytes / metabolism

Substances

  • HIF1A protein, human
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • IL1B protein, human
  • Interleukin-1beta
  • Lipopolysaccharides
  • Mannosephosphates
  • mannose-6-phosphate
  • Mannose