Fostamatinib is an effective second-line therapy in patients with immune thrombocytopenia

Br J Haematol. 2020 Sep;190(6):933-938. doi: 10.1111/bjh.16959. Epub 2020 Jul 23.

Abstract

Fostamatinib demonstrated efficacy in phase 3 trials of adults with immune thrombocytopenia (ITP). Post hoc analysis compared patients who received fostamatinib as second-line therapy (after steroids ± immunoglobulins) versus third-or-later-line therapy (after ≥2 prior lines of therapy including a second-line agent). Platelet responses ≥50 000/µl were observed in 25/32 (78%) second-line and 54/113 (48%) third-or-later-line patients. Bleeding events were less frequent in second-line (28%) versus third-or-later-line (45%) patients. Responses once achieved tended to be durable in both groups. The safety profile was similar in both groups. In this post hoc analysis, fostamatinib was more effective as second-line than third-or-later-line therapy for ITP.

Keywords: SYK; autoimmune; idiopathic thrombocytopenic purpura; platelet; spleen tyrosine kinase.

Publication types

  • Clinical Trial, Phase III
  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Aminopyridines
  • Female
  • Humans
  • Male
  • Middle Aged
  • Morpholines
  • Oxazines / administration & dosage*
  • Oxazines / adverse effects
  • Platelet Count
  • Purpura, Thrombocytopenic, Idiopathic / blood*
  • Purpura, Thrombocytopenic, Idiopathic / drug therapy*
  • Pyridines / administration & dosage*
  • Pyridines / adverse effects
  • Pyrimidines

Substances

  • Aminopyridines
  • Morpholines
  • Oxazines
  • Pyridines
  • Pyrimidines
  • fostamatinib

Grants and funding