Sch 36605, a novel anti-inflammatory compound. Taxonomy, fermentation, isolation and biological properties

J Antibiot (Tokyo). 1988 Jan;41(1):20-4. doi: 10.7164/antibiotics.41.20.

Abstract

A novel anti-inflammatory compound, Sch 36605, belonging to the blasticidin family of nucleoside compounds was isolated from the fermentation filtrate of a Streptomyces sp. Sch 36605, as well as blasticidin S, demonstrated anti-inflammatory activity in the reverse passive Arthus reaction and the adjuvant arthritic rat at doses ranging between 1-10 mg/kg and 0.3-6.0 mg/kg, respectively. A minor component, Sch 366606, co-produced in the in the fermentation was isolated and identified as a known compound in the blasticidin family of compounds.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / isolation & purification*
  • Anti-Inflammatory Agents / pharmacology
  • Fermentation
  • Guanidines / pharmacology
  • Mice
  • Nucleosides / isolation & purification*
  • Nucleosides / pharmacology
  • Rats
  • Streptomyces / classification*
  • Streptomyces / metabolism

Substances

  • Anti-Inflammatory Agents
  • Guanidines
  • Nucleosides
  • Sch 36605
  • blasticidin S