Cerium oxide nanoparticle delivery of microRNA-146a for local treatment of acute lung injury

Nanomedicine. 2021 Jun:34:102388. doi: 10.1016/j.nano.2021.102388. Epub 2021 Mar 20.

Abstract

Acute respiratory distress syndrome (ARDS) is a devastating pulmonary disease with significant in-hospital mortality and is the leading cause of death in COVID-19 patients. Excessive leukocyte recruitment, unregulated inflammation, and resultant fibrosis contribute to poor ARDS outcomes. Nanoparticle technology with cerium oxide nanoparticles (CNP) offers a mechanism by which unstable therapeutics such as the anti-inflammatory microRNA-146a can be locally delivered to the injured lung without systemic uptake. In this study, we evaluated the potential of the radical scavenging CNP conjugated to microRNA-146a (termed CNP-miR146a) in preventing acute lung injury (ALI) following exposure to bleomycin. We have found that intratracheal delivery of CNP-miR146a increases pulmonary levels of miR146a without systemic increases, and prevents ALI by altering leukocyte recruitment, reducing inflammation and oxidative stress, and decreasing collagen deposition, ultimately improving pulmonary biomechanics.

Keywords: Acute lung injury; Acute respiratory distress syndrome; Cerium oxide nanoparticles (CNP); microRNA-146a (miR146a).

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bleomycin / adverse effects*
  • Bleomycin / pharmacology
  • COVID-19 / genetics
  • COVID-19 / metabolism
  • COVID-19 Drug Treatment
  • Cerium* / chemistry
  • Cerium* / pharmacology
  • Disease Models, Animal
  • Drug Delivery Systems*
  • Male
  • Mice
  • MicroRNAs* / chemistry
  • MicroRNAs* / pharmacology
  • Respiratory Distress Syndrome / chemically induced
  • Respiratory Distress Syndrome / drug therapy*
  • Respiratory Distress Syndrome / genetics
  • Respiratory Distress Syndrome / metabolism
  • SARS-CoV-2 / metabolism

Substances

  • MicroRNAs
  • Mirn146 microRNA, mouse
  • Bleomycin
  • Cerium
  • ceric oxide