Metabolic Fate and Cardiometabolic Effects of Phenolic Compounds from Red-Fleshed Apple in Hypercholesterolemic Rats: A Comparative Study with Common White-Fleshed Apple. The AppleCOR Study

Mol Nutr Food Res. 2021 May;65(10):e2001225. doi: 10.1002/mnfr.202001225. Epub 2021 May 3.

Abstract

The present study aims to investigate the metabolic fate and the cardiometabolic effects of phenolic compounds provided by a red-fleshed apple variety biofortified in anthocyanins (ACN). Wistar rats are fed with high-fat diet (HFD) to induce hypercholesterolemia and supplemented with red-fleshed apple (HFD+R), white-fleshed apple (HFD+W), or an ACN-rich infusion from aronia fruit (HFD+A) providing matched content and profile of ACN. Plasma biochemical parameters, histological analysis, and phenol biological metabolites are determined. Plasma, urine, and feces show a significant increase of ACN metabolites after HFD+R and HFD+A, while flavan-3-ols are significantly increased after HFD+W and dihydrochalcones derivatives increased after both apples supplementation. A cardioprotective effect is observed after both apples and aronia infusion supplementation in the reduction of aortic thickness. The kidney function is improved after all supplementations and a decrease in insulin plasma concentration after both apples supplementation (HFD+R and HFD+W) is also observed. The findings support that ACN without apple matrix can induce cardioprotective effects. ACN or flavan-3-ols, together with dihydrochalcones, compose a phenolic phytocomplex in red- and white-fleshed apples, respectively, which can act synergistically in the attenuation of cardiovascular outcomes in hypercholesterolemic rats.

Keywords: Bowman's space; UPLC-MS/MS; anthocyanins; aortic thickness; phenolic compounds; red-fleshed apple; sustained intake.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anthocyanins / administration & dosage
  • Anthocyanins / pharmacokinetics
  • Cardiotonic Agents*
  • Drug Synergism
  • Female
  • Flavonoids / administration & dosage
  • Fruit / chemistry*
  • Hypercholesterolemia / drug therapy*
  • Male
  • Malus*
  • Phenols / administration & dosage*
  • Phenols / pharmacokinetics*
  • Photinia
  • Plant Extracts / administration & dosage
  • Rats
  • Rats, Wistar
  • Species Specificity

Substances

  • Anthocyanins
  • Cardiotonic Agents
  • Flavonoids
  • Phenols
  • Plant Extracts
  • flavan-3-ol