T217-Phosphorylation Exacerbates Tau Pathologies and Tau-Induced Cognitive Impairment

J Alzheimers Dis. 2021;81(4):1403-1418. doi: 10.3233/JAD-210297.

Abstract

Background: Recent studies show that an increased T217-phosphorylation of tau in plasma could diagnose AD at an early stage with high accuracy and high specificity, while the potential toxic role of tau T217-phosphorylation is not known.

Objective: To study the potential toxic role of tau T217-phosphorylation.

Methods: We performed stereotactic brain injection, behavioral testing, immunohistochemistry and immunofluorescence, western blotting, Golgi staining, in vitro recombinant tau polymerization, and other measurements.

Results: We first constructed tau T217-wild-type (T217), T217-phospho-mimic (T217E), and T217-non-phospho-mimic (T217A) plasmids or their virus vectors on the basis of wild-type tau. We found that expressing tau-T217E induced a significantly increased tau phosphorylation at multiple AD-associated sites with inhibited proteolysis and increased cleavage/fibrillization of tau, while expressing tau-T217A abolished the above changes of tau both in vitro and in vivo. By mutating T217E on tau-P301L, a dominant mutation identified in patients with frontotemporal dementia, we did not observe significant exacerbation of tau-P301L phosphorylation and cognitive impairment although the increased tau cleavage and propagation were shown.

Conclusion: T217-phosphorylation exacerbates wild-type tau hyperphosphorylation with aggravated tau cleavage/fibrillization and cognitive impairments, while overexpressing T217E on the basis P301L does not exacerbate tau phosphorylation or the P301L-induced cognitive deficits, although it aggravates tau cleavage and propagation.

Keywords: Alzheimer’s disease; T217-phosphorylation; cognition; propagation; tau.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cognition / physiology*
  • Cognitive Dysfunction / metabolism*
  • Cognitive Dysfunction / pathology
  • Hippocampus / metabolism*
  • Hippocampus / pathology
  • Humans
  • Maze Learning / physiology*
  • Mice
  • Phosphorylation
  • Tauopathies / metabolism*
  • Tauopathies / pathology
  • tau Proteins / metabolism*

Substances

  • tau Proteins