Can 68Ga-PSMA PET/CT-derived prostate-specific membrane antigen expression parameters predict prostate-specific antigen response to enzalutamide treatment?

Nucl Med Commun. 2021 Sep 1;42(9):1011-1016. doi: 10.1097/MNM.0000000000001431.

Abstract

Objective: In patients with metastatic castration-resistant prostate cancer (mCRPCa), enzalutamide is administered when docetaxel treatment fails. The purpose of the study was to evaluate the relationship between prostate-specific antigen (PSA) response and metabolic parameters obtained from 68Ga-PSMA PET/CT before treatment in this patient group.

Methods: From February 2018 to May 2020, 34 patients with mCRPCa were enrolled in this study. The association between PSA response (at least 50% decrease compared to the pretreatment value) and quantitative prostate-specific membrane antigen (PSMA) expression parameters such as SUVmax, SUVmean, PSMA-TV (PSMA receptor-expressing tumor volume) and TL-PSMA (total lesion PSMA receptor expression) were evaluated.

Results: Mean SUVmax, SUVmean, PSMA receptor-expressing tumor volume (PSMA-TV) and total lesion PSMA receptor expression (TL-PSMA) values were 33.66 ± 20.42; 8.82 ± 5.03; 319.85 ± 615.12 cm3; and 2894.76 ± 5195.13, respectively. In the posttreatment 12th week, 22 patients (64.7%) had PSA response, while 12 patients (35.3%) were nonresponders. In patients with PSA response, PSMA-TV values were significantly lower than nonresponders (78.37 ± 80.99 cm3 vs. 451.58 ± 734.61 cm3; P = 0.028). But there was no significant difference between responders and nonresponders in terms of age, ISUP grade, SUVmax, SUVmean, TL-PSMA, pretreatment PSA values, presence of local recurrence or metastases at any site.

Conclusion: PSMA-TV values on 68Ga-PSMA PET/CT imaging before starting enzalutamide treatment following docetaxel failure can predict PSA response in patients with mCRPCa.

MeSH terms

  • Aged
  • Aged, 80 and over
  • Antigens, Surface* / metabolism
  • Benzamides*
  • Edetic Acid* / analogs & derivatives
  • Gallium Isotopes*
  • Gallium Radioisotopes*
  • Glutamate Carboxypeptidase II* / metabolism
  • Humans
  • Male
  • Middle Aged
  • Nitriles* / therapeutic use
  • Oligopeptides
  • Phenylthiohydantoin* / analogs & derivatives
  • Phenylthiohydantoin* / pharmacology
  • Phenylthiohydantoin* / therapeutic use
  • Positron Emission Tomography Computed Tomography*
  • Prostate-Specific Antigen* / blood
  • Prostate-Specific Antigen* / metabolism
  • Prostatic Neoplasms, Castration-Resistant* / diagnostic imaging
  • Prostatic Neoplasms, Castration-Resistant* / drug therapy
  • Prostatic Neoplasms, Castration-Resistant* / metabolism
  • Retrospective Studies
  • Treatment Outcome

Substances

  • Nitriles
  • Gallium Isotopes
  • Prostate-Specific Antigen
  • gallium 68 PSMA-11
  • Gallium Radioisotopes
  • Phenylthiohydantoin
  • enzalutamide
  • Edetic Acid
  • Glutamate Carboxypeptidase II
  • Benzamides
  • Antigens, Surface
  • FOLH1 protein, human
  • Oligopeptides