JunD, not c-Jun, is the AP-1 transcription factor required for Ras-induced lung cancer

JCI Insight. 2021 Jul 8;6(13):e124985. doi: 10.1172/jci.insight.124985.

Abstract

The AP-1 transcription factor c-Jun is required for Ras-driven tumorigenesis in many tissues and is considered as a classical proto-oncogene. To determine the requirement for c-Jun in a mouse model of K-RasG12D-induced lung adenocarcinoma, we inducibly deleted c-Jun in the adult lung. Surprisingly, we found that inactivation of c-Jun, or mutation of its JNK phosphorylation sites, actually increased lung tumor burden. Mechanistically, we found that protein levels of the Jun family member JunD were increased in the absence of c-Jun. In c-Jun-deficient cells, JunD phosphorylation was increased, and expression of a dominant-active JNKK2-JNK1 transgene further increased lung tumor formation. Strikingly, deletion of JunD completely abolished Ras-driven lung tumorigenesis. This work identifies JunD, not c-Jun, as the crucial substrate of JNK signaling and oncogene required for Ras-induced lung cancer.

Keywords: Cell Biology; Lung cancer; Oncology.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenocarcinoma of Lung* / genetics
  • Adenocarcinoma of Lung* / metabolism
  • Animals
  • Carcinogenesis* / genetics
  • Carcinogenesis* / metabolism
  • Gene Expression Regulation, Neoplastic / genetics
  • Gene Silencing
  • Genes, jun / genetics
  • Lung Neoplasms* / genetics
  • Lung Neoplasms* / metabolism
  • MAP Kinase Kinase 7 / genetics
  • MAP Kinase Kinase 7 / metabolism
  • MAP Kinase Signaling System
  • Mice
  • Phosphorylation
  • Proto-Oncogene Proteins c-jun / genetics
  • Proto-Oncogene Proteins c-jun / metabolism*
  • Transcription Factor AP-1 / metabolism
  • ras Proteins / metabolism*

Substances

  • Proto-Oncogene Proteins c-jun
  • Transcription Factor AP-1
  • junD protein, mouse
  • MAP Kinase Kinase 7
  • Map2k7 protein, mouse
  • ras Proteins