Flavonoid glycosides from the fruits of Embelia ribes and their anti-oxidant and α-glucosidase inhibitory activities

J Asian Nat Prod Res. 2021 Aug;23(8):724-730. doi: 10.1080/10286020.2020.1776266. Epub 2020 Jun 17.

Abstract

Three new flavonoid glycosides, embeliaflavosides A-C (1-3), together with eight known flavonoid glycosides (4-11), were isolated from the fruits of Embelia ribes. Their structures were established based on the analyses of spectroscopic data. Compounds 1-11 were evaluated for antioxidant and α-glucosidase inhibitory activities. The results revealed that compounds 1-11 owned significant ABTS radical scavenging activity with IC50 values of 2.52-9.78 µM, and DPPH scavenging activity with IC50 values of 7.56-26.47 µM, respectively. However, α-glucosidase inhibition assay indicated that all the isolates were inactive.[Formula: see text].

Keywords: Embelia ribes; antioxidant activity; flavonoid glycosides; α-glucosidase inhibitory activity.

MeSH terms

  • Antioxidants / pharmacology
  • Embelia* / metabolism
  • Flavonoids / pharmacology
  • Fruit
  • Glycoside Hydrolase Inhibitors / pharmacology
  • Glycosides / pharmacology
  • Molecular Structure
  • Plant Extracts
  • Ribes* / metabolism
  • alpha-Glucosidases / metabolism

Substances

  • Antioxidants
  • Flavonoids
  • Glycoside Hydrolase Inhibitors
  • Glycosides
  • Plant Extracts
  • alpha-Glucosidases