Copper-Mediated Cross-Coupling of Diazo Compounds with Sulfinates

Org Lett. 2021 Sep 3;23(17):6919-6924. doi: 10.1021/acs.orglett.1c02481. Epub 2021 Aug 19.

Abstract

A copper-mediated cross-coupling reaction between a diazo compound and a sodium alkane(arene)sulfinate gives a sulfone as the product. This reaction proceeds under mild conditions and features excellent functional group compatibility. A wide range of sodium alkane(arene)sulfinates were successfully applied in this chemistry. Mechanistic studies revealed that the overall reaction efficiency of the sulfinates was in line with their nucleophilicity in this reaction.

Publication types

  • Research Support, Non-U.S. Gov't