One new phenylpropanoid glycoside from Myxopyrum smilacifolium with α-glucosidase inhibitory activity

J Asian Nat Prod Res. 2022 Sep;24(9):891-897. doi: 10.1080/10286020.2021.1992392. Epub 2021 Nov 25.

Abstract

One new phenylpropanoid glycoside, myxosmoside I (1) and six known compounds, arenarioside (2), verbacoside (3), 3-formylindole (4), 5-hydroxymethyl furfural (5), D-manitol (6), and glycerol monooleate (7) were isolated from the roots of Myxopyrum smilacifolium (Wall.) Blume. Their chemical structures were determined by 1D-, 2D-NMR, and mass spectra, chemical methods, and compared with those reported in the literature. All compounds were evaluated for α-glucosidase inhibitory effect. Among them, phenylpropanoid glycosides 1-3 significantly inhibited α-glucosidase activity with IC50 values of 30.0 ± 0.9, 66.6 ± 2.3, and 36.9 ± 2.0 µM, respectively.

Keywords: Myxopyrum smilacifolium; Oleaceae; myxosmoside; phenylpropanoid glycoside; α-glucosidase.

MeSH terms

  • Cardiac Glycosides*
  • Glycoside Hydrolase Inhibitors / chemistry
  • Glycoside Hydrolase Inhibitors / pharmacology
  • Glycosides / chemistry
  • Glycosides / pharmacology
  • Molecular Structure
  • Oleaceae*
  • alpha-Glucosidases

Substances

  • Cardiac Glycosides
  • Glycoside Hydrolase Inhibitors
  • Glycosides
  • alpha-Glucosidases