A Cell-Based Platform for the Investigation of Immunoproteasome Subunit β5i Expression and Biology of β5i-Containing Proteasomes

Cells. 2021 Nov 5;10(11):3049. doi: 10.3390/cells10113049.

Abstract

The degradation of most intracellular proteins is a dynamic and tightly regulated process performed by proteasomes. To date, different forms of proteasomes have been identified. Currently the role of non-constitutive proteasomes (immunoproteasomes (iPs) and intermediate proteasomes (intPs)) has attracted special attention. Here, using a CRISPR-Cas9 nickase technology, four cell lines: histiocytic lymphoma, colorectal adenocarcinoma, cervix adenocarcinoma, and hepatocarcinoma were modified to express proteasomes with mCherry-tagged β5i subunit, which is a catalytic subunit of iPs and intPs. Importantly, the expression of the chimeric gene in modified cells is under the control of endogenous regulatory mechanisms and is increased following IFN-γ and/or TNF-α stimulation. Fluorescent proteasomes retain catalytic activity and are distributed within the nucleus and cytoplasm. RNAseq reveals marginal differences in gene expression profiles between the modified and wild-type cell lines. Predominant metabolic pathways and patterns of expressed receptors were identified for each cell line. Using established cell lines, we demonstrated that anti-cancer drugs Ruxolitinib, Vincristine and Gefitinib stimulated the expression of β5i-containing proteasomes, which might affect disease prognosis. Taken together, obtained cell lines can be used as a platform for real-time studies of immunoproteasome gene expression, localization of iPs and intPs, interaction of non-constitutive proteasomes with other proteins, proteasome trafficking and many other aspects of proteasome biology in living cells. Moreover, the established platform might be especially useful for fast and large-scale experiments intended to evaluate the effects of different conditions including treatment with various drugs and compounds on the proteasome pool.

Keywords: immunoproteasome; intermediate proteasome; non-constitutive proteasome; proteasome; reporter cell line.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / pharmacology
  • Cell Line, Tumor
  • Cell Nucleus / drug effects
  • Cell Nucleus / metabolism
  • Fluorescence
  • Gefitinib / pharmacology
  • Gene Expression Regulation, Neoplastic / drug effects
  • Genome, Human
  • Humans
  • Interferon-gamma / pharmacology
  • Nitriles / pharmacology
  • Proteasome Endopeptidase Complex / immunology*
  • Protein Subunits / metabolism*
  • Pyrazoles / pharmacology
  • Pyrimidines / pharmacology
  • Tumor Necrosis Factor-alpha / pharmacology
  • Vincristine / pharmacology

Substances

  • Antineoplastic Agents
  • Nitriles
  • Protein Subunits
  • Pyrazoles
  • Pyrimidines
  • Tumor Necrosis Factor-alpha
  • Vincristine
  • Interferon-gamma
  • ruxolitinib
  • Proteasome Endopeptidase Complex
  • Gefitinib