Alpha-terpineol grafted acetylated lentinan as an anti-bacterial adhesion agent

Carbohydr Polym. 2022 Feb 1:277:118825. doi: 10.1016/j.carbpol.2021.118825. Epub 2021 Oct 29.

Abstract

Biomedical implants-associated bacterial infections have become a major threat to human health. Therefore, it is meaningful to develop new antibacterial strategies to solve this problem. In this study, we conjugated acetylated lentinan (AceLNT) with α-terpineol (AceLNT-g-α-ter), a highly effective natural antibacterial compound, to constitute a novel AceLNT-g-α-ter membrane (AceLNT-g-α-terM). Compared with AceLNT membrane (AceLNTM), the adhesion amount of E. coli and P. aeruginosa in AceLNT-g-α-terM decreased by 80% and 85% after 7 d incubation in fluid bacterial medium. Moreover, the number of E. coli and P. aeruginosa biofilm on AceLNT-g-α-terM surface decreased by 70% and 71%. At the meanwhile, α-terpineol grafting modification of AceLNT had limited effect on its stimulating activity on macrophages and had no more cytotoxicity. In summary, our study firstly confirmed that AceLNT-g-α-terM could effectively inhibit gram-negative bacteria adhesion and biofilm formation, and provided a novel strategy for preventing infection of biomedical implants.

Keywords: Acetylated lentinan; Anti-bacterial adhesion; Anti-biofilm; α-terpineol.

MeSH terms

  • Acetylation
  • Animals
  • Anti-Bacterial Agents / chemical synthesis
  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / pharmacology*
  • Bacterial Adhesion / drug effects
  • Biofilms / drug effects
  • Cyclohexane Monoterpenes / chemistry
  • Cyclohexane Monoterpenes / pharmacology*
  • Cytokines / metabolism
  • Escherichia coli / drug effects*
  • Lentinan / chemistry
  • Lentinan / pharmacology*
  • Macrophages / drug effects
  • Macrophages / metabolism
  • Mice
  • Microbial Sensitivity Tests
  • Molecular Structure
  • NIH 3T3 Cells
  • Pseudomonas aeruginosa / drug effects*
  • RAW 264.7 Cells
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Anti-Bacterial Agents
  • Cyclohexane Monoterpenes
  • Cytokines
  • Tumor Necrosis Factor-alpha
  • alpha-terpineol
  • Lentinan