Hippocampal BMP signaling as a common pathway for antidepressant action

Cell Mol Life Sci. 2021 Dec 22;79(1):31. doi: 10.1007/s00018-021-04026-y.

Abstract

The benefits of current treatments for depression are limited by low response rates, delayed therapeutic effects, and multiple side effects. Antidepressants affect a variety of neurotransmitter systems in different areas of the brain, and the mechanisms underlying their convergent effects on behavior have been unclear. Here we identify hippocampal bone morphogenetic protein (BMP) signaling as a common downstream pathway that mediates the behavioral effects of five different antidepressant classes (fluoxetine, bupropion, duloxetine, vilazodone, trazodone) and of electroconvulsive therapy. All of these therapies decrease BMP signaling and enhance neurogenesis in the hippocampus. Preventing the decrease in BMP signaling blocks the effect of antidepressant treatment on behavioral phenotypes. Further, inhibition of BMP signaling in hippocampal newborn neurons is sufficient to produce an antidepressant effect, while chemogenetic silencing of newborn neurons prevents the antidepressant effect. Thus, inhibition of hippocampal BMP signaling is both necessary and sufficient to mediate the effects of multiple classes of antidepressants.

Keywords: Adult neurogenesis; Antidepressants; BMP signaling; Depression.

MeSH terms

  • Aging / pathology
  • Animals
  • Anti-Anxiety Agents / pharmacology
  • Antidepressive Agents / pharmacology*
  • Behavior, Animal / drug effects
  • Bone Morphogenetic Proteins / metabolism*
  • Dentate Gyrus / drug effects
  • Dentate Gyrus / metabolism
  • Duloxetine Hydrochloride / pharmacology
  • Electroconvulsive Therapy
  • Fluoxetine / pharmacology
  • Ganglia, Spinal / drug effects
  • Ganglia, Spinal / pathology
  • Hippocampus / drug effects
  • Hippocampus / metabolism*
  • Mice
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Neurogenesis / drug effects
  • Signal Transduction* / drug effects
  • Stress, Psychological / complications
  • Trazodone / pharmacology
  • Vilazodone Hydrochloride / pharmacology

Substances

  • Anti-Anxiety Agents
  • Antidepressive Agents
  • Bone Morphogenetic Proteins
  • Fluoxetine
  • Duloxetine Hydrochloride
  • Vilazodone Hydrochloride
  • Trazodone