Noncoding genetic variation in GATA3 increases acute lymphoblastic leukemia risk through local and global changes in chromatin conformation

Nat Genet. 2022 Feb;54(2):170-179. doi: 10.1038/s41588-021-00993-x. Epub 2022 Feb 3.

Abstract

Inherited noncoding genetic variants confer significant disease susceptibility to childhood acute lymphoblastic leukemia (ALL) but the molecular processes linking germline polymorphisms with somatic lesions in this cancer are poorly understood. Through targeted sequencing in 5,008 patients, we identified a key regulatory germline variant in GATA3 associated with Philadelphia chromosome-like ALL (Ph-like ALL). Using CRISPR-Cas9 editing and samples from patients with Ph-like ALL, we showed that this variant activated a strong enhancer that upregulated GATA3 transcription. This, in turn, reshaped global chromatin accessibility and three-dimensional genome organization, including regions proximal to the ALL oncogene CRLF2. Finally, we showed that GATA3 directly regulated CRLF2 and potentiated the JAK-STAT oncogenic effects during leukemogenesis. Taken together, we provide evidence for a distinct mechanism by which a germline noncoding variant contributes to oncogene activation, epigenetic regulation and three-dimensional genome reprogramming.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Child
  • Chromatin / chemistry*
  • Chromatin / metabolism
  • Enhancer Elements, Genetic
  • Female
  • GATA3 Transcription Factor / genetics*
  • GATA3 Transcription Factor / metabolism
  • Genetic Predisposition to Disease*
  • Genome, Human
  • Humans
  • Janus Kinases / metabolism
  • Male
  • Oncogenes
  • Philadelphia Chromosome
  • Polymorphism, Single Nucleotide*
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma / genetics*
  • Protein Binding
  • Receptors, Cytokine / genetics
  • Receptors, Cytokine / metabolism
  • STAT Transcription Factors / metabolism
  • Signal Transduction
  • Up-Regulation

Substances

  • CRLF2 protein, human
  • Chromatin
  • GATA3 Transcription Factor
  • GATA3 protein, human
  • Receptors, Cytokine
  • STAT Transcription Factors
  • Janus Kinases