Anomeric Thioglycosides Give Different Anomeric Product Distributions under NIS/TfOH Activation

J Org Chem. 2022 Mar 18;87(6):4154-4167. doi: 10.1021/acs.joc.1c03001. Epub 2022 Mar 3.

Abstract

The reaction of a series of anomeric thioglycosides with various glycosyl acceptors and N-iodosuccinimide/catalytic triflic acid was investigated with respect to reactivity and anomeric selectivity. In general, β-configured donors were found to give a more β-selective reaction outcome compared to their α-configured counterparts. The relative reactivity of various thioglycosides was measured through competition experiments, and the following order was established: phenyl, tolyl, methyl, ethyl, isopropyl, and 1-adamantyl.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Catalysis
  • Glycosylation
  • Thioglycosides*

Substances

  • Thioglycosides