The pyrogenic actions of the interferon-inducer, polyinosinic:polycytidylic acid are antagonised by ketoprofen

Eur J Pharmacol. 1987 Jun 4;137(2-3):257-60. doi: 10.1016/0014-2999(87)90231-7.

Abstract

The effect of various doses of polyinosinic:polycytidilic acid (Poly I:C) in the range (0.25-250 micrograms/kg) administered i.v. on the body temperature of rabbits was investigated. The effect of ketoprofen on the febrile responses was also studied. The threshold dose of Poly I:C administered which produced a fever was between 0.25 and 0.5 micrograms/kg and a double-sigmoidal dose-response relationship was observed. A sigmoidal relationship was obtained with lower doses from 0.25 micrograms/kg to an apparent maximum with 2.5 micrograms/kg and another with higher doses from 5 micrograms/kg to another apparent maximum with 250 micrograms/kg. Ketoprofen (3 mg/kg) given s.c. 15 min prior to Poly I:C inhibited the production of fever. Ketoprofen administered after the onset of fever resulted in an immediate deffervescence. These results suggest that febrile responses to Poly I:C involve prostaglandin biosynthesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Injections, Intravenous
  • Ketoprofen / pharmacology*
  • Male
  • Phenylpropionates / pharmacology*
  • Poly I-C / antagonists & inhibitors*
  • Poly I-C / toxicity
  • Pyrogens / antagonists & inhibitors*
  • Rabbits

Substances

  • Phenylpropionates
  • Pyrogens
  • Ketoprofen
  • Poly I-C