In vitro and in vivo evidence that the switch from calcineurin to mTOR inhibitors may be a strategy for immunosuppression in Epstein-Barr virus-associated post-transplant lymphoproliferative disorder

Kidney Int. 2022 Dec;102(6):1392-1408. doi: 10.1016/j.kint.2022.08.025. Epub 2022 Sep 11.

Abstract

Post-transplant lymphoproliferative disorder is a life-threatening complication of immunosuppression following transplantation mediated by failure of T cells to control Epstein-Barr virus (EBV)-infected and transformed B cells. Typically, a modification or reduction of immunosuppression is recommended, but insufficiently defined thus far. In order to help delineate this, we characterized EBV-antigen-specific T cells and lymphoblastoid cell lines from healthy donors and in patients with a kidney transplant in the absence or presence of the standard immunosuppressants tacrolimus, cyclosporin A, prednisolone, rapamycin, and mycophenolic acid. Phenotypes of lymphoblastoid cell-lines and T cells, T cell-receptor-repertoire diversity, and T-cell reactivity upon co-culture with autologous lymphoblastoid cell lines were analyzed. Rapamycin and mycophenolic acid inhibited lymphoblastoid cell-line proliferation. T cells treated with prednisolone and rapamycin showed nearly normal cytokine production. Proliferation and the viability of T cells were decreased by mycophenolic acid, while tacrolimus and cyclosporin A were strong suppressors of T-cell function including their killing activity. Overall, our study provides a basis for the clinical decision for the modification and reduction of immunosuppression and adds information to the complex balance of maintaining anti-viral immunity while preventing acute rejection. Thus, an immunosuppressive regime based on mTOR inhibition and reduced or withdrawn calcineurin inhibitors could be a promising strategy for patients with increased risk of or manifested EBV-associated post-transplant lymphoproliferative disorder.

Keywords: Epstein–Barr virus; T cells; calcineurin inhibitors; immunosuppression; lymphoblastoid cell lines; mycophenolic acid; post-transplant lymphoproliferative disorder; rapamycin; transplantation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcineurin / genetics
  • Cyclosporine / pharmacology
  • Cyclosporine / therapeutic use
  • Epstein-Barr Virus Infections* / drug therapy
  • Herpesvirus 4, Human
  • Humans
  • Immunosuppression Therapy
  • Immunosuppressive Agents / therapeutic use
  • Lymphoproliferative Disorders* / drug therapy
  • Lymphoproliferative Disorders* / etiology
  • Lymphoproliferative Disorders* / prevention & control
  • MTOR Inhibitors
  • Mycophenolic Acid / therapeutic use
  • Prednisolone / pharmacology
  • Prednisolone / therapeutic use
  • Sirolimus / pharmacology
  • Sirolimus / therapeutic use
  • TOR Serine-Threonine Kinases
  • Tacrolimus / pharmacology
  • Tacrolimus / therapeutic use

Substances

  • Tacrolimus
  • Calcineurin
  • MTOR Inhibitors
  • Cyclosporine
  • Mycophenolic Acid
  • Immunosuppressive Agents
  • Sirolimus
  • Prednisolone
  • MTOR protein, human
  • TOR Serine-Threonine Kinases