Ketone Body Infusion Abrogates Growth Hormone-Induced Lipolysis and Insulin Resistance

J Clin Endocrinol Metab. 2023 Feb 15;108(3):653-664. doi: 10.1210/clinem/dgac595.

Abstract

Context: Exogenous ketone body administration lowers circulating glucose levels but the underlying mechanisms are uncertain.

Objective: We tested the hypothesis that administration of the ketone body β-hydroxybutyrate (βOHB) acutely increases insulin sensitivity via feedback suppression of circulating free fatty acid (FFA) levels.

Methods: In a randomized, single-blinded crossover design, 8 healthy men were studied twice with a growth hormone (GH) infusion to induce lipolysis in combination with infusion of either βOHB or saline. Each study day comprised a basal period and a hyperinsulinemic-euglycemic clamp combined with a glucose tracer and adipose tissue and skeletal muscle biopsies.

Results: βOHB administration profoundly suppressed FFA levels concomitantly with a significant increase in glucose disposal and energy expenditure. This was accompanied by a many-fold increase in skeletal muscle content of both βOHB and its derivative acetoacetate.

Conclusion: Our data unravel an insulin-sensitizing effect of βOHB, which we suggest is mediated by concomitant suppression of lipolysis.

Trial registration: ClinicalTrials.gov NCT02655263.

Keywords: free fatty acids; glucose metabolism; growth hormone; insulin sensitivity; ketone bodies; β-hydroxybutyrate.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3-Hydroxybutyric Acid / pharmacology
  • Fatty Acids, Nonesterified
  • Glucose
  • Glucose Clamp Technique
  • Growth Hormone
  • Human Growth Hormone* / pharmacology
  • Humans
  • Insulin / pharmacology
  • Insulin Resistance* / physiology
  • Ketone Bodies* / pharmacology
  • Ketone Bodies* / therapeutic use
  • Lipolysis / drug effects
  • Lipolysis / physiology
  • Male

Substances

  • 3-Hydroxybutyric Acid
  • Fatty Acids, Nonesterified
  • Glucose
  • Growth Hormone
  • Human Growth Hormone
  • Insulin
  • Ketone Bodies

Associated data

  • ClinicalTrials.gov/NCT02655263