Brief Report: Effect of Antiretroviral Switch From Tenofovir Disoproxil fumarate to Tenofovir Alafenamide on Alanine Aminotransferase, Lipid Profiles, and Renal Function in HIV/HBV-Coinfected Individuals in a Nationwide Canadian Study

J Acquir Immune Defic Syndr. 2022 Dec 1;91(4):368-372. doi: 10.1097/QAI.0000000000003079.

Abstract

Objective: Tenofovir alafenamide (TAF) achieves increased renal safety and improved alanine aminotransferase (ALT) normalization but increased lipid profile in hepatitis B virus (HBV)-monoinfected patients switched from tenofovir disoproxil fumarate (TDF). It is unclear whether HIV coinfection perturbs these biochemical changes. To this end, we assessed these parameters in HIV/HBV-coinfected patients switched from TDF to TAF.

Design: Retrospective, multicenter, observational study.

Methods: HIV/HBV-coinfected patients switched from TDF to TAF-based antiretroviral therapy (ART) at 6 Canadian Hepatitis B Network (CanHepB) academic sites were included. Changes in lipid profile, estimated glomerular filtration rate (eGFR), and ALT were evaluated using linear mixed effect model regression.

Results: Eighty-two HIV/HBV-coinfected patients with a mean 103-week follow-up duration were identified. At time of TAF switch, 80 of 82 (98%) were HBV virally suppressed, 29 of 82 (35%) had elevated ALT levels, and 63 of 82 (77%) had eGFR of ≥60 mL/min per 1.73 m 2 . Twenty-six/Eighty-two (32%) had preexisting renal comorbidities. There were no changes in total cholesterol, high-density lipoprotein, low-density lipoprotein, and triglyceride levels 2 years after TAF switch. Those with elevated ALT levels achieved greater ALT normalization after TAF switch (-0.004 [-0.008 to 0.0] log 10 U/L/mo, P = 0.03). eGFR decline rate while on TDF (-0.66 [-0.23 to -1.08] mL/min/month, P < 0.005) was diminished after switching to TAF (-0.02 [-0.16 to 0.11] mL/min/mo, P = 0.7) and those with eGFR of <60 mL/min experienced increase in eGFR after TAF switch (0.45 [0.03-0.87] mL/min/mo, P = 0.04).

Conclusions: Our study supports switching from TDF to TAF with positive influence on overall long-term biochemical profile in HIV/HBV-coinfected individuals.

Publication types

  • Observational Study
  • Multicenter Study

MeSH terms

  • Adenine / therapeutic use
  • Alanine / therapeutic use
  • Alanine Transaminase
  • Anti-Retroviral Agents / therapeutic use
  • Canada
  • Cholesterol
  • Coinfection*
  • HIV Infections* / complications
  • HIV Infections* / drug therapy
  • Hepatitis B virus
  • Humans
  • Kidney / physiology
  • Lipids
  • Lipoproteins, HDL
  • Lipoproteins, LDL
  • Retrospective Studies
  • Tenofovir / therapeutic use
  • Triglycerides

Substances

  • Tenofovir
  • Alanine Transaminase
  • Alanine
  • Adenine
  • Anti-Retroviral Agents
  • Lipids
  • Cholesterol
  • Lipoproteins, HDL
  • Triglycerides
  • Lipoproteins, LDL