First-line treatments for patients with advanced ALK gene rearrangements in NSCLC: a systematic review and network meta-analysis

J Int Med Res. 2022 Nov;50(11):3000605221132703. doi: 10.1177/03000605221132703.

Abstract

Objective: To conduct a network meta-analysis of randomised controlled trials to determine the optimal clinical choice of first-line therapy for patients with ALK receptor tyrosine kinase (ALK) gene rearrangement non-small cell lung cancer (NSCLC).

Methods: Clinical trials in patients with histologically confirmed ALK gene rearrangement NSCLC, that included ALK inhibitors as first-line therapy, were identified using database searches. A Bayesian network meta-analysis was conducted to calculate the efficacy and safety of the included first-line treatments.

Results: Nine trials with 2,407 patients were included for analyses. Lorlatinib was better than brigatinib for progression-free survival (PFS) (hazard ratio 0.79, 95% confidence interval 0.63, 0.98). In subgroup analyses, lorlatinib exhibited the highest probability of best PFS ranking in patients with or without baseline brain metastases (38% and 80%, respectively); brigatinib had the highest probability of best PFS ranking among Asian patients (47%). Alectinib offered the highest survival advantage (57% probability), while lorlatinib was likely to be the best treatment for an objective response (41% probability). Alectinib displayed the highest probability of being ranked lowest for grade ≥3 adverse events (86%).

Conclusions: Lorlatinib was associated with the best PFS overall, and was suitable for patients with or without brain metastases. Brigatinib was associated with the best PFS in Asian patients.

Keywords: ALK inhibitors; Non-small cell lung cancer; anaplastic lymphoma kinase; brigatinib; first-line therapy; lorlatinib.

Publication types

  • Meta-Analysis
  • Systematic Review

MeSH terms

  • Anaplastic Lymphoma Kinase / genetics
  • Bayes Theorem
  • Brain Neoplasms* / drug therapy
  • Brain Neoplasms* / genetics
  • Carcinoma, Non-Small-Cell Lung* / drug therapy
  • Carcinoma, Non-Small-Cell Lung* / genetics
  • Carcinoma, Non-Small-Cell Lung* / pathology
  • Gene Rearrangement
  • Humans
  • Lactams, Macrocyclic / adverse effects
  • Lung Neoplasms* / drug therapy
  • Lung Neoplasms* / genetics
  • Lung Neoplasms* / pathology
  • Network Meta-Analysis
  • Protein Kinase Inhibitors / adverse effects
  • Randomized Controlled Trials as Topic

Substances

  • Anaplastic Lymphoma Kinase
  • brigatinib
  • Lactams, Macrocyclic
  • lorlatinib
  • Protein Kinase Inhibitors