Dose of ibrutinib in Waldenström macroglobulinaemia: Less can be more

Br J Haematol. 2023 Jun;201(5):807-808. doi: 10.1111/bjh.18664. Epub 2023 Jan 30.

Abstract

Ibrutinib changed the landscape of treatment in Waldenström macroglobulinaemia (WM) with excellent responses; however, there are high rates of dose reduction due to adverse events. The impact of this reduced dosing is unclear with regards to outcomes. Sarosiek and colleagues provide valuable data in a very large retrospective study demonstrating that dose reduction is effective in managing adverse events in the majority, with equivalent, if not better, outcomes than those without dose reductions.

Keywords: Waldenstrom macroglobulinaemia; bruton tyrosine kinase inhibitor; ibrutinib.

MeSH terms

  • Humans
  • Protein Kinase Inhibitors* / pharmacology
  • Protein Kinase Inhibitors* / therapeutic use
  • Pyrazoles / adverse effects
  • Pyrimidines / therapeutic use
  • Retrospective Studies
  • Waldenstrom Macroglobulinemia* / drug therapy

Substances

  • ibrutinib
  • Pyrazoles
  • Pyrimidines
  • Protein Kinase Inhibitors