Electrophysiologic properties of falipamil (AQA-39)--a new bradycardiac agent

Eur Heart J. 1987 Nov;8(11):1236-40. doi: 10.1093/oxfordjournals.eurheartj.a062198.

Abstract

Falipamil hydrochloride (AQA 39) is a new antiarrhythmic agent structurally related to verapamil. We evaluated the electrophysiologic properties of intravenous falipamil (1.5 mg kg-1 within 20 minutes) in 12 patients. The spontaneous cycle length was significantly (P less than 0.001) prolonged (+79 +/- 59 ms). Atrioventricular conduction was significantly (P less than 0.001) shorter due to AH interval shortening (-17 +/- 14 ms), most probably related to an anticholinergic effect. Similarly, the anterograde Wenckebach point occurred at a significantly (P less than 0.06) higher rate after falipamil (+10 +/- 7 beats min-1). No statistically significant effect was noted on the refractory periods of the AV node, although there was a trend to shortening. The refractoriness of the right atrium and ventricle was significantly prolonged. It is concluded that falipamil is a bradycardiac agent with electrophysiologic properties quite different from those of verapamil and similar to those of class IA antiarrhythmic agents.

MeSH terms

  • Aged
  • Anti-Arrhythmia Agents*
  • Atrioventricular Node / drug effects
  • Coronary Disease / physiopathology
  • Electrophysiology
  • Female
  • Heart / drug effects*
  • Heart Atria / drug effects
  • Heart Rate / drug effects
  • Heart Ventricles / drug effects
  • Humans
  • Isoindoles
  • Male
  • Middle Aged
  • Phthalimides / pharmacology*

Substances

  • Anti-Arrhythmia Agents
  • Isoindoles
  • Phthalimides
  • falipamil