PD-1/PD-L1 immune checkpoint blockade in ovarian cancer: Dilemmas and opportunities

Drug Discov Today. 2023 Aug;28(8):103666. doi: 10.1016/j.drudis.2023.103666. Epub 2023 Jun 9.

Abstract

Immune checkpoint inhibitors (ICIs) have revolutionized treatment in oncology. Antibodies against PD-1/PD-L1 and ICI-based combinations are under clinical investigations in multiple cancers, including ovarian cancer. However, the success of ICIs has not materialized in ovarian cancer, which remains one of the few malignancies where ICIs exhibit modest efficacy as either monotherapy or combination therapy. In this review, we summarize completed and ongoing clinical trials of PD-1/PD-L1 blockade in ovarian cancer, categorize the underlying mechanisms of resistance emergence, and introduce candidate approaches to rewire the tumor microenvironment (TME) to potentiate anti-PD-1/PD-L1 antibodies.

Keywords: PD-1/PD-L1 blockade; drug resistance; immune checkpoint inhibitors; ovarian cancer.

Publication types

  • Review
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies
  • B7-H1 Antigen
  • Combined Modality Therapy
  • Female
  • Humans
  • Immune Checkpoint Inhibitors* / pharmacology
  • Immune Checkpoint Inhibitors* / therapeutic use
  • Ovarian Neoplasms* / drug therapy
  • Tumor Microenvironment

Substances

  • Immune Checkpoint Inhibitors
  • B7-H1 Antigen
  • Antibodies