Effect of sulpiride on amphetamine-induced behaviour in relation to changes in striatal dopamine release in vivo

Eur J Pharmacol. 1986 Oct 7;129(3):411-5. doi: 10.1016/0014-2999(86)90459-0.

Abstract

Intracerebral dialysis was used to simultaneously monitor extracellular dopamine (DA) in striatum and behaviour in rats following administration of amphetamine and sulpiride. Amphetamine (2 mg/kg s.c.) caused a marked release of DA into striatal perfusates, an effect which was potentiated in rats pretreated with sulpiride (50 mg/kg s.c.). Amphetamine-induced stereotyped head and forepaw movements were potentiated by sulpiride at a time point corresponding with the enhanced release of DA. In comparison, amphetamine-induced locomotor activity was completely inhibited by sulpiride.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Behavior, Animal / drug effects*
  • Corpus Striatum / drug effects
  • Corpus Striatum / metabolism
  • Dextroamphetamine / pharmacology*
  • Dopamine / metabolism*
  • Male
  • Motor Activity / drug effects
  • Rats
  • Rats, Inbred Strains
  • Stereotyped Behavior / drug effects
  • Sulpiride / pharmacology*

Substances

  • Sulpiride
  • Dextroamphetamine
  • Dopamine