Acquired resistance to crizotinib in novel CDK14-ALK and CLTC-ALK fusions of ALK-positive large B-cell lymphoma identified by next-generation sequencing

Cancer Biol Ther. 2023 Dec 31;24(1):2271212. doi: 10.1080/15384047.2023.2271212. Epub 2023 Oct 31.

Abstract

Anaplastic lymphoma kinase-positive large B-cell lymphoma (ALK+ LBCL) is a rare subtype of non-Hodgkin lymphoma. ALK inhibitors are being tried to treat recurrent/refractory ALK+ LBCL. A majority of patients with ALK+ tumors respond to crizotinib, but partial cases ultimately develop resistance about a year later. Here, we report a case of ALK+ LBCL carrying a new fusion gene involving CDK14 and ALK, CLTC-ALK gene rearrangements and MTOR gene mutation. The patient had progressive disease after combination of crizotinib and chemotherapy treatment about 5.5 months later, accompanied by reduced abundance of CDK14-ALK, increased abundance of CLTC-ALK and a novel MFHAS1 gene mutation. However, MTOR mutation turned negative. The patient received alectinib combined with hyper-CVAD, then followed by alectinib as monotherapy for 21 months. The patient achieved partial response and remained in a stable condition. This case suggests that CDK14-ALK fusion gene may be more sensitive to crizotinib than CLTC-ALK fusion gene. MTOR is associated with the anti-tumor mechanism of ALK inhibitors. MFHAS1 gene mutation and/or CLTC-ALK gene copy number amplification may involve resistance to crizotinib. Furthermore, alectinib may inhibit the carcinogenicity of these gene changes and improve the prognosis of ALK+ LBCL.

Keywords: ALK; CDK14; CLTC; MFHAS1; crizotinib; large B-cell lymphoma.

Plain language summary

The novel CDK14-ALK fusion gene in ALK+ LBCL was sensitive to crizotinib.MFHAS1 gene mutation and/or CLTC-ALK gene copy number amplification may involve resistance to crizotinib.

Publication types

  • Case Reports
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anaplastic Lymphoma Kinase / genetics
  • Carbazoles / pharmacology
  • Carbazoles / therapeutic use
  • Carcinoma, Non-Small-Cell Lung* / pathology
  • Cell Cycle Proteins / genetics
  • Crizotinib / pharmacology
  • Crizotinib / therapeutic use
  • DNA-Binding Proteins / genetics
  • Drug Resistance, Neoplasm / genetics
  • High-Throughput Nucleotide Sequencing
  • Humans
  • Lung Neoplasms* / pathology
  • Lymphoma, B-Cell* / drug therapy
  • Mutation
  • Oncogene Proteins / genetics
  • Protein Kinase Inhibitors / pharmacology
  • Protein Kinase Inhibitors / therapeutic use
  • TOR Serine-Threonine Kinases / genetics

Substances

  • Anaplastic Lymphoma Kinase
  • Carbazoles
  • CDK14 protein, human
  • Cell Cycle Proteins
  • CLTC protein, human
  • Crizotinib
  • DNA-Binding Proteins
  • MFHAS1 protein, human
  • Oncogene Proteins
  • Protein Kinase Inhibitors
  • TOR Serine-Threonine Kinases

Grants and funding

81470347/National Natural Science Foundation of China.