[Compounds with potential antitumor activity. V. 2-Substituted 3-[2-(1,3,4-thiadazolyl)]-4-thiazolidinone]

Farmaco Sci. 1986 Nov;41(11):839-51.
[Article in Italian]

Abstract

The synthesis of a series of 2-substituted 3-[2-(1,3,4-thiadiazolyl)]-4-thiazolidinones is described. Evaluation of these derivatives against P 388 lymphocytic leukemia growth in mice revealed that no compound shows significant activity. 2-(2-Thienyl)-3-[2-(1,3,4-thiadiazolyl)]-4-thiazolidinone (I) whose significant activity on P 388 leukemia was reported in a previous paper, was tested against other experimental tumors: it exhibits slight activity also against L 1210 leukemia and M 5076 ascitic sarcoma.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Antineoplastic Agents / chemical synthesis*
  • Leukemia L1210 / drug therapy
  • Leukemia P388 / drug therapy
  • Mice
  • Sarcoma, Experimental / drug therapy
  • Thiadiazoles / chemical synthesis*
  • Thiadiazoles / pharmacology
  • Thiazoles / chemical synthesis*
  • Thiazoles / pharmacology

Substances

  • Antineoplastic Agents
  • Thiadiazoles
  • Thiazoles