Triptolide inhibits the proinflammatory potential of myeloid-derived suppressor cells via reducing Arginase-1 in rheumatoid arthritis

Int Immunopharmacol. 2024 Jan 25:127:111345. doi: 10.1016/j.intimp.2023.111345. Epub 2023 Dec 11.

Abstract

Triptolide (TPT) is widely used in the treatment of rheumatoid arthritis (RA). However, its regulatory mechanisms are not fully understood. This study demonstrated that Myeloid-derived suppressor cells (MDSCs) were expanded in both RA patients and arthritic mice. The frequency of MDSCs was correlated with RA disease severity and T helper 17 (Th17) responses. MDSCs from RA patients promoted the polarization of Th17 cells in vitro, which could be substantially attenuated by blocking arginase-1 (Arg-1). TPT inhibited the differentiation of MDSCs, particularly the monocytic MDSCs (M-MDSCs) subsets, as well as the expression of Arg-1 in a dose dependent manner. Alongside, TPT treatment reduced the potential of MDSCs to promote the polarization of IL-17+ T cell in vitro. Consistently, TPT immunotherapy alleviated adjuvant-induced arthritis (AIA) in a mice model, and reduced the frequency of MDSCs, M-MDSCs and IL-17+ T cells simultaneously. The presented data suggest a pathogenic role of MDSCs in RA and may function as a novel and effective therapeutic target for TPT in RA.

Keywords: Arginase-1; Myeloid-derived suppressor cells; Rheumatoid arthritis; Th17 cells; Triptolide.

MeSH terms

  • Animals
  • Arginase / metabolism
  • Arthritis, Rheumatoid* / metabolism
  • Diterpenes*
  • Epoxy Compounds
  • Humans
  • Interleukin-17 / metabolism
  • Mice
  • Myeloid-Derived Suppressor Cells* / metabolism
  • Phenanthrenes*

Substances

  • Interleukin-17
  • triptolide
  • Arginase
  • Diterpenes
  • Epoxy Compounds
  • Phenanthrenes