Inhibition of voluntary ethanol intake in rats by a combination of dihydroergotoxine and thioridazine

Alcohol Drug Res. 1987;7(4):285-90.

Abstract

Dihydroergotoxine (DHET) decreased voluntary ethanol intake in rats selected for their stable ethanol preference (mean daily ethanol intake 8 g/kg). DHET inhibition was markedly potentiated by thioridazine. The potentiation is explained with a synergistic inhibitory effect on dopaminergic transmission: that is, DHET acting on dopamine (DA) autoreceptors and thioridazine preferentially inhibiting postsynaptic DA receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alcohol Drinking / drug effects*
  • Animals
  • Dihydroergotoxine / pharmacology*
  • Dopamine Antagonists
  • Drug Synergism
  • Inhibition, Psychological
  • Male
  • Rats
  • Rats, Inbred Strains
  • Receptors, Dopamine / drug effects
  • Thioridazine / pharmacology*

Substances

  • Dopamine Antagonists
  • Receptors, Dopamine
  • Dihydroergotoxine
  • Thioridazine