Three-year outcomes of valoctocogene roxaparvovec gene therapy for hemophilia A

J Thromb Haemost. 2024 Jul;22(7):1880-1893. doi: 10.1016/j.jtha.2024.04.001. Epub 2024 Apr 12.

Abstract

Background: Valoctocogene roxaparvovec transfers a human factor (F)VIII coding sequence into hepatocytes of people with severe hemophilia A to provide bleeding protection.

Objectives: To present 3-year efficacy and safety in the multicenter, open-label, single-arm, phase 3 GENEr8-1 trial.

Methods: GENEr8-1 enrolled 134 adult males with severe hemophilia A who were receiving FVIII prophylaxis. Efficacy endpoints included annualized bleeding rate, annualized FVIII utilization, FVIII activity (chromogenic substrate assay; imputed as 1 IU/dL at baseline and 0 IU/dL after discontinuation), and the Haemophilia-Specific Quality of Life Questionnaire for Adults. Safety was assessed by adverse events (AEs).

Results: At week 156, 131 of 134 participants remained in the study; overall, 17 of 134 resumed prophylaxis. Mean annualized bleeding rate for treated bleeds decreased from 4.8 (SD, 6.5) bleeds/y at baseline to 0.8 (SD, 2.3; P < .0001) bleeds/y after prophylaxis (prophylaxis cessation to last follow-up) and 0.97 (SD, 3.48) bleeds/y during year 3. Annualized FVIII utilization decreased 96.8% from baseline after prophylaxis and 94.2% during year 3. At week 156, mean and median FVIII activity were 18.4 (SD, 30.8) and 8.3 IU/dL, respectively. FVIII activity decrease was lower between years 2 and 3 than between years 1 and 2. At the end of year 3, clinically meaningful improvements in the Haemophilia-Specific Quality of Life Questionnaire for Adults Total Score were observed (mean change from baseline, 6.6; 95% CI, 4.24-8.87; P < .0001). Mild alanine aminotransferase elevations remained the most common AE during year 3 (23.7% of participants). A serious AE of B-cell acute lymphoblastic leukemia was considered unrelated to treatment.

Conclusion: Hemostatic efficacy was maintained, and safety remained unchanged from previous years.

Keywords: adeno-associated virus; clinical trial; gene therapy; health-related quality of life; hemophilia A; phase 3.

Publication types

  • Multicenter Study
  • Clinical Trial, Phase III

MeSH terms

  • Adolescent
  • Adult
  • Coagulants / adverse effects
  • Coagulants / therapeutic use
  • Factor VIII* / adverse effects
  • Factor VIII* / genetics
  • Factor VIII* / therapeutic use
  • Genetic Therapy*
  • Hemophilia A* / blood
  • Hemophilia A* / drug therapy
  • Hemophilia A* / genetics
  • Hemophilia A* / therapy
  • Hemorrhage*
  • Hepatocytes
  • Humans
  • Male
  • Middle Aged
  • Quality of Life*
  • Surveys and Questionnaires
  • Time Factors
  • Treatment Outcome
  • Young Adult

Substances

  • Factor VIII
  • F8 protein, human
  • Coagulants