Eicosapentaenoic acid-mediated activation of PGAM2 regulates skeletal muscle growth and development via the PI3K/AKT pathway

Int J Biol Macromol. 2024 May;268(Pt 2):131547. doi: 10.1016/j.ijbiomac.2024.131547. Epub 2024 Apr 17.

Abstract

Eicosapentaenoic acid regulates glucose uptake in skeletal muscle and significantly affects whole-body energy metabolism. However, the underlying molecular mechanism remains unclear. Here we report that eicosapentaenoic acid activates phosphoglycerate mutase 2, which mediates the conversion of 2-phosphoglycerate into 3-phosphoglycerate. This enzyme plays a pivotal role in glycerol degradation, thereby facilitating the proliferation and differentiation of satellite cells in skeletal muscle. Interestingly, phosphoglycerate mutase 2 inhibits mitochondrial metabolism, promoting the formation of fast-type muscle fibers. Treatment with eicosapentaenoic acid and phosphoglycerate mutase 2 knockdown induced opposite transcriptomic changes, most of which were enriched in the PI3K-AKT signaling pathway. Phosphoglycerate mutase 2 activated the PI3K-AKT signaling pathway, which inhibited the phosphorylation of FOXO1, and, in turn, inhibited mitochondrial function and promoted the formation of fast-type muscle fibers. Our results suggest that eicosapentaenoic acid promotes skeletal muscle growth and regulates glucose metabolism by targeting phosphoglycerate mutase 2 and activating the PI3K/AKT signaling pathway.

Keywords: Eicosapentaenoic acid; Mitochondria; Muscle fiber type transformation; Myogenesis; Phosphoglycerate mutase 2.

MeSH terms

  • Animals
  • Cell Differentiation / drug effects
  • Cell Proliferation / drug effects
  • Eicosapentaenoic Acid* / pharmacology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mitochondria / drug effects
  • Mitochondria / metabolism
  • Muscle Development / drug effects
  • Muscle, Skeletal* / drug effects
  • Muscle, Skeletal* / metabolism
  • Phosphatidylinositol 3-Kinases* / metabolism
  • Phosphoglycerate Mutase / genetics
  • Phosphoglycerate Mutase / metabolism
  • Proto-Oncogene Proteins c-akt* / metabolism
  • Signal Transduction* / drug effects
  • Swine

Substances

  • Eicosapentaenoic Acid
  • Phosphatidylinositol 3-Kinases
  • Phosphoglycerate Mutase
  • Proto-Oncogene Proteins c-akt