Pharmacological characterization of sex differences in the effects of dopaminergic drugs on effort-based decision making in rats

Psychopharmacology (Berl). 2024 Oct;241(10):2033-2044. doi: 10.1007/s00213-024-06615-8. Epub 2024 Jun 6.

Abstract

Rationale: Motivational dysfunctions related to effort exertion are common in psychiatric disorders. Dopamine systems regulate exertion of effort and effort-based choice in humans and rodents.

Objectives: Previous rodent studies mainly employed male rats, and it is imperative to conduct studies in male and female rats.

Methods: The present studies compared the effort-related effects of IP injections of the dopamine antagonists ecopipam and haloperidol, and the vesicular monoamine transport-2 inhibitor tetrabenazine (TBZ), in male and female rats using the fixed ratio 5/chow feeding choice task.

Results: Ecopipam (0.05-0.2 mg/kg) and haloperidol (0.05-0.15 mg/kg) induced a low-effort bias, decreasing lever pressing and increasing chow intake in males and females in the same dose range. With lever pressing, there was a modest but significant dose x sex interaction after ecopipam injection, but there was no significant interaction after administration of haloperidol. In the first study with TBZ (0.25-1.0 mg/kg), there was a robust sex difference. TBZ shifted choice from lever pressing to chow intake in male rats, but was ineffective in females. In a second experiment, 2.0 mg/kg affected choice behavior in both males and females. TBZ increased accumbens c-Fos immunoreactivity in a sex-dependent manner, with males significantly increasing at 1.0 mg/kg, while females showed augmented immunoreactivity at 2.0 mg/kg.

Conclusions: The neural and behavioral effects of TBZ differed across sexes, emphasizing the importance of conducting studies in male and female rats. This research has implications for understanding the effort-related motivational dysfunctions seen in psychopathology.

Keywords: Anergia; Avolition; Behavioral activation; Choice; Fatigue; Motivation.

MeSH terms

  • Animals
  • Benzazepines
  • Choice Behavior / drug effects
  • Decision Making / drug effects
  • Dopamine Antagonists* / administration & dosage
  • Dopamine Antagonists* / pharmacology
  • Dose-Response Relationship, Drug*
  • Female
  • Haloperidol* / pharmacology
  • Male
  • Motivation / drug effects
  • Nucleus Accumbens / drug effects
  • Nucleus Accumbens / metabolism
  • Proto-Oncogene Proteins c-fos / metabolism
  • Rats
  • Rats, Sprague-Dawley
  • Sex Characteristics
  • Tetrabenazine* / administration & dosage
  • Tetrabenazine* / pharmacology

Substances

  • Haloperidol
  • Dopamine Antagonists
  • Tetrabenazine
  • ecopipam
  • Proto-Oncogene Proteins c-fos
  • Benzazepines