Expression of a kinase inactive SLK is embryonic lethal and impairs cell migration in fibroblasts

Biochim Biophys Acta Mol Cell Res. 2024 Oct;1871(7):119783. doi: 10.1016/j.bbamcr.2024.119783. Epub 2024 Jun 12.

Abstract

Kinases are known to have kinase activity independent functions. To gain further insights into potential kinase-independent functions of SLK/STK2, we have developed a kinase-dead allele, SLKK63R using in vivo CRISPR/Cas technology. Our studies show that blastocysts homozygote for SLKK63R do not develop into viable mice. However, heterozygotes are viable and fertile with no overt phenotypes. Analyses of mouse embryonic fibroblasts show that expression of SLKK63R results in a 50% decrease in kinase activity in heterozygotes. In contrast to previous studies, our data show that SLK does not form homodimers and that the kinase defective allele does not act in a dominant negative fashion. Expression of SLKK63R leads to altered Rac1 and RhoA activity, increased stress fiber formation and delayed focal adhesion turnover. Our data support a previously observed role for SLK in cell migration and suggest that at least 50% kinase activity is sufficient for embryonic development.

Keywords: Kinase inactive; Migration; SLK; Ste20-like kinase; Stk2.

MeSH terms

  • Animals
  • CRISPR-Cas Systems
  • Cell Movement* / genetics
  • Embryo Loss / genetics
  • Embryo Loss / pathology
  • Embryo, Mammalian / cytology
  • Embryo, Mammalian / metabolism
  • Female
  • Fibroblasts* / cytology
  • Fibroblasts* / metabolism
  • Focal Adhesions / genetics
  • Focal Adhesions / metabolism
  • Mice
  • Neuropeptides
  • Protein Serine-Threonine Kinases* / genetics
  • Protein Serine-Threonine Kinases* / metabolism
  • rac1 GTP-Binding Protein* / genetics
  • rac1 GTP-Binding Protein* / metabolism
  • rhoA GTP-Binding Protein / genetics
  • rhoA GTP-Binding Protein / metabolism

Substances

  • Neuropeptides
  • Protein Serine-Threonine Kinases
  • rac1 GTP-Binding Protein
  • Rac1 protein, mouse
  • rhoA GTP-Binding Protein
  • RhoA protein, mouse
  • SLK protein, mouse