Therapeutic potential of co-signaling receptor modulation in hepatitis B

Cell. 2024 Jul 25;187(15):4078-4094.e21. doi: 10.1016/j.cell.2024.05.038. Epub 2024 Jun 18.

Abstract

Reversing CD8+ T cell dysfunction is crucial in treating chronic hepatitis B virus (HBV) infection, yet specific molecular targets remain unclear. Our study analyzed co-signaling receptors during hepatocellular priming and traced the trajectory and fate of dysfunctional HBV-specific CD8+ T cells. Early on, these cells upregulate PD-1, CTLA-4, LAG-3, OX40, 4-1BB, and ICOS. While blocking co-inhibitory receptors had minimal effect, activating 4-1BB and OX40 converted them into antiviral effectors. Prolonged stimulation led to a self-renewing, long-lived, heterogeneous population with a unique transcriptional profile. This includes dysfunctional progenitor/stem-like (TSL) cells and two distinct dysfunctional tissue-resident memory (TRM) populations. While 4-1BB expression is ubiquitously maintained, OX40 expression is limited to TSL. In chronic settings, only 4-1BB stimulation conferred antiviral activity. In HBeAg+ chronic patients, 4-1BB activation showed the highest potential to rejuvenate dysfunctional CD8+ T cells. Targeting all dysfunctional T cells, rather than only stem-like precursors, holds promise for treating chronic HBV infection.

Keywords: 4-1BB; CD8(+) T cells; OX40; T cell dysfunction; chronic viral infection; hepatitis B virus; immunotherapy; liver.

MeSH terms

  • Animals
  • Antigens, CD / metabolism
  • CD8-Positive T-Lymphocytes* / immunology
  • CD8-Positive T-Lymphocytes* / metabolism
  • Hepatitis B virus*
  • Hepatitis B, Chronic* / drug therapy
  • Hepatitis B, Chronic* / metabolism
  • Hepatitis B, Chronic* / virology
  • Humans
  • Mice
  • Programmed Cell Death 1 Receptor / metabolism
  • Receptors, OX40 / metabolism
  • Signal Transduction
  • Tumor Necrosis Factor Receptor Superfamily, Member 9 / metabolism

Substances

  • Tumor Necrosis Factor Receptor Superfamily, Member 9
  • Receptors, OX40
  • Programmed Cell Death 1 Receptor
  • Antigens, CD