Ursodeoxycholic acid and COVID-19 outcomes: a cohort study and data synthesis of state-of-art evidence

Expert Rev Anti Infect Ther. 2024 Dec;22(12):1239-1250. doi: 10.1080/14787210.2024.2376153. Epub 2024 Jul 9.

Abstract

Background: The potential of ursodeoxycholic acid (UDCA) in inhibiting angiotensin-converting enzyme 2 was demonstrated. However, conflicting evidence emerged regarding the association between UDCA and COVID-19 outcomes, prompting the need for a comprehensive investigation.

Research design and methods: Patients diagnosed with COVID-19 infection were retrospectively analyzed and divided into two groups: the UDCA-treated group and the control group. Kaplan-Meier recovery analysis and Cox proportional hazards models were used to evaluate the recovery time and hazard ratios. Additionally, study-level pooled analyses for multiple clinical outcomes were performed.

Results: In the 115-patient cohort, UDCA treatment was significantly associated with a reduced recovery time. The subgroup analysis suggests that the 300 mg subgroup had a significant (adjusted hazard ratio: 1.63 [95% CI, 1.01 to 2.60]) benefit with a shorter duration of fever. The results of pooled analyses also show that UDCA treatment can significantly reduce the incidence of severe/critical diseases in COVID-19 (adjusted odds ratio: 0.68 [95% CI, 0.50 to 0.94]).

Conclusions: UDCA treatment notably improves the recovery time following an Omicron strain infection without observed safety concerns. These promising results advocate for UDCA as a viable treatment for COVID-19, paving the way for further large-scale and prospective research to explore the full potential of UDCA.

Keywords: COVID-19; Ursodeoxycholic acid; cohort study; data synthesis; retrospective study.

MeSH terms

  • Adult
  • Aged
  • Betacoronavirus / drug effects
  • COVID-19 Drug Treatment
  • COVID-19*
  • Cholagogues and Choleretics / administration & dosage
  • Cholagogues and Choleretics / therapeutic use
  • Cohort Studies
  • Female
  • Humans
  • Kaplan-Meier Estimate
  • Male
  • Middle Aged
  • Pandemics
  • Pneumonia, Viral / drug therapy
  • Proportional Hazards Models
  • Retrospective Studies
  • SARS-CoV-2* / drug effects
  • Treatment Outcome
  • Ursodeoxycholic Acid* / administration & dosage
  • Ursodeoxycholic Acid* / therapeutic use

Substances

  • Ursodeoxycholic Acid
  • Cholagogues and Choleretics