Store-operated calcium entry dysfunction in CRAC channelopathy: Insights from a novel STIM1 mutation

Clin Immunol. 2024 Aug:265:110306. doi: 10.1016/j.clim.2024.110306. Epub 2024 Jul 6.

Abstract

Store-operated calcium entry (SOCE) plays a crucial role in maintaining cellular calcium homeostasis. This mechanism involves proteins, such as stromal interaction molecule 1 (STIM1) and ORAI1. Mutations in the genes encoding these proteins, especially STIM1, can lead to various diseases, including CRAC channelopathies associated with severe combined immunodeficiency. Herein, we describe a novel homozygous mutation, NM_003156 c.792-3C > G, in STIM1 in a patient with a clinical profile of CRAC channelopathy, including immune system deficiencies and muscle weakness. Functional analyses revealed three distinct spliced forms in the patient cells: wild-type, exon 7 skipping, and intronic retention. Calcium influx analysis revealed impaired SOCE in the patient cells, indicating a loss of STIM1 function. We developed an antisense oligonucleotide treatment that improves STIM1 splicing and highlighted its potential as a therapeutic approach. Our findings provide insights into the complex effects of STIM1 mutations and shed light on the multifaceted clinical presentation of the patient.

Keywords: CRAC channelopathy; Immunodeficiency; STIM1; Splicing; Store-operated calcium entry; Therapy.

Publication types

  • Case Reports

MeSH terms

  • Calcium Release Activated Calcium Channels / genetics
  • Calcium Release Activated Calcium Channels / metabolism
  • Calcium* / metabolism
  • Channelopathies / genetics
  • Female
  • Humans
  • Male
  • Mutation*
  • Neoplasm Proteins* / genetics
  • Neoplasm Proteins* / metabolism
  • ORAI1 Protein / genetics
  • ORAI1 Protein / metabolism
  • Severe Combined Immunodeficiency / genetics
  • Stromal Interaction Molecule 1* / genetics
  • Stromal Interaction Molecule 1* / metabolism

Substances

  • Stromal Interaction Molecule 1
  • STIM1 protein, human
  • Neoplasm Proteins
  • Calcium
  • Calcium Release Activated Calcium Channels
  • ORAI1 Protein