Digoxin is still useful, but is still causing toxicity

Cleve Clin J Med. 2024 Aug 1;91(8):489-499. doi: 10.3949/ccjm.91a.23105.

Abstract

Digoxin, the oldest known cardiovascular drug, is still used today to treat heart failure and atrial fibrillation. Because it has a narrow therapeutic index and multiple interactions, it frequently causes toxicity with a wide range of symptoms and cardiac arrhythmias. More importantly, elevated serum digoxin levels have been linked to a higher risk of death in patients with heart failure or atrial fibrillation, even without signs or symptoms of toxicity. This article reviews the current state of digoxin use, its pharmacologic principles, and the mechanisms, clinical presentation, and management of toxicity.

Publication types

  • Review

MeSH terms

  • Anti-Arrhythmia Agents / adverse effects
  • Atrial Fibrillation* / drug therapy
  • Cardiotonic Agents / adverse effects
  • Cardiotonic Agents / pharmacology
  • Cardiotonic Agents / therapeutic use
  • Digoxin* / adverse effects
  • Digoxin* / blood
  • Heart Failure* / chemically induced
  • Humans

Substances

  • Digoxin
  • Cardiotonic Agents
  • Anti-Arrhythmia Agents