Novel pesticides design: co-encapsulation of citral and cyproconazole for the control of Botrytis cinerea using biocompatible nano-carriers

Pest Manag Sci. 2024 Dec;80(12):6096-6106. doi: 10.1002/ps.8337. Epub 2024 Aug 2.

Abstract

Background: Growing concerns about sustainability have driven the search for eco-friendly pest management solutions. Combining natural and synthetic compounds within controlled release systems is a promising strategy. This study investigated the co-encapsulation of the natural compound citral (Cit) and the synthetic antifungal cyproconazole (CPZ) using two water-based nanocarriers: solid lipid nanoparticles (SLNs) and chitosan nanoparticles (CSNPs).

Results: Both CSNPs and SLNs loaded with Cit + CPZ displayed superior antifungal activity against Botrytis cinerea compared to free compounds. Notably, CSNPs with a 2:1 Cit:CPZ ratio exhibited the highest efficacy, achieving a minimum inhibitory concentration (MIC100) of < 1.56 μg mL-1, lower than the 12.5 μg mL-1 of non-encapsulated compounds. This formulation significantly reduced the required synthetic CPZ while maintaining efficacy, highlighting its potential for environmentally friendly pest control.

Conclusion: The successful co-encapsulation of Cit + CPZ within CSNPs, particularly at a 2:1 ratio, demonstrates a promising approach for developing effective and sustainable antifungal formulations against B. cinerea. © 2024 Society of Chemical Industry.

Keywords: Botrytis cinerea; citral; cyproconazole; nanoencapsulated; nano‐carriers; novel antifungal.

MeSH terms

  • Acyclic Monoterpenes* / pharmacology
  • Antifungal Agents / chemistry
  • Antifungal Agents / pharmacology
  • Botrytis* / drug effects
  • Chitosan / chemistry
  • Chitosan / pharmacology
  • Drug Carriers / chemistry
  • Drug Compounding
  • Fungicides, Industrial* / chemistry
  • Fungicides, Industrial* / pharmacology
  • Lipids / chemistry
  • Microbial Sensitivity Tests
  • Nanoparticles* / chemistry
  • Plant Diseases / microbiology
  • Plant Diseases / prevention & control
  • Triazoles / chemistry
  • Triazoles / pharmacology

Substances

  • citral
  • Acyclic Monoterpenes
  • Fungicides, Industrial
  • Triazoles
  • Chitosan
  • Drug Carriers
  • Antifungal Agents
  • Lipids

Supplementary concepts

  • Botrytis cinerea