Adiponectin receptor agonist AdipoRon alleviates memory impairment in the hippocampus of septic mice

Behav Brain Res. 2024 Aug 24:472:115174. doi: 10.1016/j.bbr.2024.115174. Epub 2024 Aug 3.

Abstract

Sepsis-associated encephalopathy (SAE) is a common and severe clinical feature of sepsis; however, therapeutic approaches are limited because of the unclear pathogenesis. Adiponectin receptor agonist (AdipoRon) is a small-molecule agonist of the adiponectin receptor that exhibits anti-inflammatory and memory-improving effects in various diseases. In the present study, we established lipopolysaccharide (LPS)-induced mice models of SAE and found that Adiponectin receptor 1 (AdipoR1) was significantly decreased in the hippocampus. Administration of AdipoRon improves memory impairment, mitigates synaptic damage, and alleviates neuronal death. Furthermore, AdipoRon reduces the number of microglia. More importantly, AdipoRon promotes the phosphorylation of adenosine 5 '-monophosphate activated protein kinase (pAMPK). In conclusion, AdipoRon is protective against SAE-induced memory decline and brain injury in the SAE models via activating the hippocampal adenosine 5 '-monophosphate activated protein kinase (AMPK).

Keywords: AMPK; AdipoRon; Memory impairment; Microglia; SAE.

MeSH terms

  • AMP-Activated Protein Kinases / metabolism
  • Animals
  • Disease Models, Animal*
  • Hippocampus* / drug effects
  • Hippocampus* / metabolism
  • Lipopolysaccharides / pharmacology
  • Male
  • Memory Disorders* / drug therapy
  • Mice
  • Mice, Inbred C57BL
  • Microglia / drug effects
  • Microglia / metabolism
  • Piperidines / pharmacology
  • Receptors, Adiponectin* / agonists
  • Receptors, Adiponectin* / metabolism
  • Sepsis / complications
  • Sepsis / drug therapy
  • Sepsis / metabolism
  • Sepsis-Associated Encephalopathy / drug therapy
  • Sepsis-Associated Encephalopathy / metabolism

Substances

  • adiponectin receptor 1, mouse
  • AdipoRon
  • AMP-Activated Protein Kinases
  • Lipopolysaccharides
  • Piperidines
  • Receptors, Adiponectin