A comprehensive gas chromatography electron ionization high resolution mass spectrometry study of a new steroidal selective androgen receptor modulator (SARM) compound S42

J Mass Spectrom. 2024 Aug;59(8):e5077. doi: 10.1002/jms.5077.

Abstract

The synthetic 20-keto-steroid S42 (1) demonstrated selective androgen receptor modulator (SARM) properties in preclinical studies and, consequently, received growing attention also in the context of sports drug testing programs. Fundamental understanding of the behavior of S42 (1) and of relevant derivatives in gas chromatography-electron ionization MS experiments at high resolution (GC-EI-HRMS) is indispensable to develop a reliable qualitative and quantitative doping control method for S42 (1) and its metabolites in body fluid matrices. We present important fundamental mechanistic data on the EI fragmentation behavior of S42 (1) and of silyl ether derivatives as well as of stable isotope-labelled reference material.

Keywords: 20‐keto steroid S42; EI‐MS fragmentation mechanisms; GC‐EI‐HRMS; silyl ether derivatives; stable isotope derivatives.

MeSH terms

  • Anabolic Agents / analysis
  • Anabolic Agents / chemistry
  • Androgens / analysis
  • Androgens / chemistry
  • Doping in Sports* / prevention & control
  • Gas Chromatography-Mass Spectrometry* / methods
  • Humans
  • Receptors, Androgen* / analysis
  • Receptors, Androgen* / chemistry
  • Receptors, Androgen* / metabolism
  • Spectrometry, Mass, Electrospray Ionization / methods
  • Steroids / analysis
  • Steroids / chemistry
  • Substance Abuse Detection / methods

Substances

  • Receptors, Androgen
  • Anabolic Agents
  • Androgens
  • Steroids