Effects of High-altitude Hypoxia on Drug Metabolism and Pharmacokinetics of Sedative-hypnotic Drugs and Regulatory Mechanism

Curr Drug Metab. 2024;25(6):416-424. doi: 10.2174/0113892002318723240802100729.

Abstract

Sedative hypnotics effectively improve sleep quality under high-altitude hypoxia by reducing central nervous system excitability. High-altitude hypoxia causes sleep disorders and modifies the metabolism and mechanisms of drug action, impacting medication therapy's effectiveness. This review aims to provide a theoretical basis for the treatment of central nervous system diseases in high-altitude areas by summarizing the progress and mechanism of sedative-hypnotics in hypoxic environments, as well as the impact of high-altitude hypoxia on sleep.

Keywords: Drug metabolism; drug transport; high-altitude hypoxia; rational use of drugs.; sedative-hypnotics; sleep disorders.

Publication types

  • Review

MeSH terms

  • Altitude
  • Altitude Sickness / drug therapy
  • Altitude Sickness / metabolism
  • Animals
  • Humans
  • Hypnotics and Sedatives* / pharmacokinetics
  • Hypoxia* / metabolism

Substances

  • Hypnotics and Sedatives